ALDH1A2-IN-1

Names

[ CAS No. ]:
2204229-64-9

[ Name ]:
ALDH1A2-IN-1

Biological Activity

[Description]:

ALDH1A2-IN-1 is an active site-directed reversible ALDH1A2 inhibitor (IC50=0.91 μM; Kd=0.26 μM) with several hydrophobic interactions[1].

[Related Catalog]:

Signaling Pathways >> Metabolic Enzyme/Protease >> Aldehyde Dehydrogenase (ALDH)

Research Areas >> Endocrinology

[Target]

IC50: 0.91 μM (ALDH1A2), Kd: 0.26 μM (ALDH1A2)[1]

[References]

[1]. Chen Y, et al. Structural Basis of ALDH1A2 Inhibition by Irreversible and Reversible Small Molecule Inhibitors. ACS Chem Biol. 2018;13(3):582-590.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₁H₂₆N₄O₄S

[ Molecular Weight ]:
430.52

Related Compounds

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