PF-4840154
Names
Biological Activity
[Description]:
PF-4840154 is a potent, selective agonist of the rat and human TrpA1 channel with EC50s of 97 and 23 nM, respectively.
[Related Catalog]:
[Target]
IC50: 97 nM (rTrpA1), 23 nM (hTrpA1)[1]
[References]
[Related Small Molecules]
capsaicin
|
Capsazepine
|
EIPA
|
Diphenyleneiodonium chloride
|
HC-030031
|
SKF-96365
|
HC 067047
|
AMG 9810
|
GSK-1016790A
|
SAR7334
|
RN-1734
|
AMG-517
|
SB-366791
|
IcilinAG-3-5
|
ML204
Chemical & Physical Properties
[ Density]:
1.2±0.1 g/cm3
[ Molecular Formula ]:
C26H38N6O2
[ Molecular Weight ]:
466.619
[ Exact Mass ]:
466.305634
[ LogP ]:
6.03
[ Index of Refraction ]:
1.589
[ Storage condition ]:
2-8℃