Alkyl, unsaturated,(hetero) aryl, and N-protected α-amino ketones by acylation of organometallic reagents

AR Katritzky, KNB Le, L Khelashvili…

Index: Herbert, John M.; Maggiani, Maria Synthetic Communications, 2001 , vol. 31, # 6 p. 947 - 951

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Citation Number: 51

Abstract

... Volume: Page: ... the presence of Et 3 N for the N-acylation of amines 3 and amides, 3,4 the O-acylation of aldehydes, 5 and the C-acylation of ketones and heteroaromatics, 6 alkylsulfones, 7 ... Figure 2 Grignard reagents and heteroaryllithium reagents (R 2 M) 2a−e ...