Naltrindole hydrochloride
Naltrindole hydrochloride structure
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Common Name | Naltrindole hydrochloride | ||
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| CAS Number | 111469-81-9 | Molecular Weight | 450.95700 | |
| Density | N/A | Boiling Point | 664.2ºC at 760mmHg | |
| Molecular Formula | C26H27ClN2O3 | Melting Point | N/A | |
| MSDS | Chinese USA | Flash Point | 355.5ºC | |
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Naltrindole, a highly selective and potent non-peptide delta opioid receptor antagonist.
Eur. J. Pharmacol. 146 , 185, (1988)
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Acute delta-opioid receptor activation induces CREB phosphorylation in NG108-15 cells.
Eur. J. Pharmacol. 390 , 1-6, (2000) A growing body of evidence supports an important role of the transcription factor cAMP responsive element binding protein (CREB) in mediating opioid-induced changes in the cAMP pathway. Regulation of CREB and subsequent changes in gene expression may underlie... |
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Characterization of delta-opioid receptors and effect of enkephalins on IRD 98 rat epithelial intestinal cell line.
Pflugers Arch. 439 , 547-554, (2000) Using 3H-Tyr-D-Ala-Gly-Phe-D-Leu-OH (3H-DADLE) as a radioligand, delta-opioid binding sites on the IRD 98 rat epithelial cell line were identified. These sites were found to be reversible, saturable, specific and displayed high affinity for DADLE. Scatchard a... |