TYR-D-ALA-GLY-PHE-D-LEU ACETATE SALT
TYR-D-ALA-GLY-PHE-D-LEU ACETATE SALT structure
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Common Name | TYR-D-ALA-GLY-PHE-D-LEU ACETATE SALT | ||
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| CAS Number | 94825-57-7 | Molecular Weight | 629.70100 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C31H43N5O9 | Melting Point | N/A | |
| MSDS | Chinese USA | Flash Point | N/A | |
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Species differences in the effects of the κ-opioid receptor antagonist zyklophin.
Alcohol 51 , 43-9, (2016) We have shown that dysregulation of the dynorphin/kappa-opioid receptor (DYN/KOR) system contributes to escalated alcohol self-administration in alcohol dependence and that KOR antagonists with extended durations of action selectively reduce escalated alcohol... |
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Delta opioid peptide [D-Ala2,D-leu5]enkephalin blocks the long-term loss of dopamine transporters induced by multiple administrations of methamphetamine: involvement of opioid receptors and reactive oxygen species.
J. Pharmacol. Exp. Ther. 287 , 322, (1998) Delta opioid peptide [D-Ala2,D-leu5]enkephalin (DADLE) can prolong organ preservation and increases myocardial tolerance to ischemia. Our study examined the protective property of DADLE against methamphetamine- (METH) induced dopaminergic terminal damage in t... |
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Mitogenic signalling by delta opioid receptors expressed in rat-1 fibroblasts involves activation of the p70s6k/p85s6k S6 kinase.
Biochem. J. 325 , 217-222, (1997) The regulation of mitogenic signalling pathways by G-protein-coupled receptors has been studied in Rat-1 fibroblasts stably transfected with the murine delta opioid receptor. We showed recently that stimulation of this receptor led to the activation of the p4... |
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Delta opioid peptide[D- Ala(2),D-Leu(5)]enkephalin promotes cell survival.
J. Biomed. Sci. 7 , 195, (2000) By studying the hibernation in ground squirrels, a protein factor termed hibernation induction trigger (HIT) was found to induce hibernation in summer-active ground squirrels. Further purification of HIT yielded an 88-kD peptide that is enriched in winter hib... |
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Gz mediates the long-lasting desensitization of brain CB1 receptors and is essential for cross-tolerance with morphine.
Mol. Psychiatry 5 , 11, (2009) Although the systemic administration of cannabinoids produces antinociception, their chronic use leads to analgesic tolerance as well as cross-tolerance to morphine. These effects are mediated by cannabinoids binding to peripheral, spinal and supraspinal CB1 ... |
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Delta opioid receptors expressed by stably transfected jurkat cells signal through the map kinase pathway in a ras-independent manner.
J. Neuroimmunol. 94 , 48-57, (1999) Delta opioid receptors (DOR) are G-protein coupled 7-transmembrane receptors (GPCR), expressed by thymic and splenic T cells, that modulate interleukin (IL)-2 production and proliferation in response to concanavalin A or crosslinking the TCR. Mitogen-activate... |