5-METHOXYGRAMINE

5-METHOXYGRAMINE Structure
5-METHOXYGRAMINE structure
Common Name 5-METHOXYGRAMINE
CAS Number 16620-52-3 Molecular Weight 204.26800
Density 1.119g/cm3 Boiling Point 334.7ºC at 760 mmHg
Molecular Formula C12H16N2O Melting Point 123-126 °C(lit.)
MSDS Chinese USA Flash Point 156.2ºC

Regulation of serotonin 5-HT2C receptors by chronic ligand exposure.

Eur. J. Pharmacol. 498(1-3) , 59-69, (2004)

The effect of ligand pretreatment on human 5-hydroxytryptamine2C (5-HT2C) receptors was examined in CHO cells expressing high (CHO-1C7; 67+/-3 pmol/mg) or low (CHO-1C19; 72+/-10 fmol/mg) levels of the receptor. Seventy-two hours pretreatment of CHO-1C7 cells ...

Kinetics of competitive drug action at 5-hydroxytryptamine2 receptors in isolated rabbit aorta.

J. Pharmacol. Exp. Ther. 242(1) , 108-14, (1987)

The kinetics of agonist and antagonist interactions with the 5-hydroxytryptamine2 receptor were studied in the isolated rabbit aorta by following the antagonist-induced decrease in the steady-state response to an agonist. A model describing the competitive dr...