TERT-BUTYL-BICYCLO [2.2.2]
![TERT-BUTYL-BICYCLO [2.2.2] Structure](https://image.chemsrc.com/caspic/095/70636-86-1.png)
TERT-BUTYL-BICYCLO [2.2.2] structure
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Common Name | TERT-BUTYL-BICYCLO [2.2.2] | ||
|---|---|---|---|---|
| CAS Number | 70636-86-1 | Molecular Weight | 222.24200 | |
| Density | 1.25g/cm3 | Boiling Point | 231.3ºC at 760 mmHg | |
| Molecular Formula | C8H15O3PS | Melting Point | N/A | |
| MSDS | USA | Flash Point | 93.7ºC | |
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J. Physiol. 590(Pt 1) , 163-78, (2012) Picrotoxin and t-butylbicyclophosphorothionate (TBPS) are GABA(A) receptor (GABA(A)R) open channel blockers. However, picrotoxin displaceable [(35)S]TBPS binding to α1β2γ2 GABA(A)Rs occurs in the absence of GABA, suggesting that access to the binding site is ... |
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A synthetic 18-norsteroid distinguishes between two neuroactive steroid binding sites on GABAA receptors.
J. Pharmacol. Exp. Ther. 333(2) , 404-13, (2010) In the absence of GABA, neuroactive steroids that enhance GABA-mediated currents modulate binding of [35S]t-butylbicyclophosphorothionate in a biphasic manner, with enhancement of binding at low concentrations (site NS1) and inhibition at higher concentration... |
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Brain regional heterogeneity of pH effects on GABA(A) receptor-associated [35s]TBPS binding.
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