Efficient and scalable method for the selective alkylation and acylation of secondary amines in the presence of primary amines

F Laduron, V Tamborowski, L Moens…

文献索引：Organic Process Research and Development, , vol. 9, # 1 p. 102 - 104

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被引用次数: 21

摘要

... 3 or benzaldehyde 4 that have to be removed after deprotection, making the process more expensive. ... (b) Green, TW; Wuts, PGM Protective Groups in Organic Synthesis, 3rd ... 1995, 36, 3451 [CrossRef], [CAS] A one-step procedure for the selective trifluoroacetylation of primary ...