Efficient and scalable method for the selective alkylation and acylation of secondary amines in the presence of primary amines

F Laduron, V Tamborowski, L Moens…

Index: Organic Process Research and Development, , vol. 9, # 1 p. 102 - 104

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Citation Number: 21

Abstract

... 3 or benzaldehyde 4 that have to be removed after deprotection, making the process more expensive. ... (b) Green, TW; Wuts, PGM Protective Groups in Organic Synthesis, 3rd ... 1995, 36, 3451 [CrossRef], [CAS] A one-step procedure for the selective trifluoroacetylation of primary ...

Palladium-mediated N-arylation of heterocyclic diamines: Ins...

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Synthesis and in vitro antibacterial activity of novel methy...

[Srivastava, Brijesh Kumar; Soni, Rina; Patel, Jayendra Z.; Solanki, Manish; Valani, Darshan; Gupta, Sunil; Mishra, Bhupendra; Takale, Vijay; Pandya, Purvi; Jain, Mukul R.; Patel, Pankaj R. Bioorganic and Medicinal Chemistry Letters, 2007 , vol. 17, # 18 p. 5227 - 5232]

Fluorine-18 labeled benzamides for studying the dopamine D2 ...

[Mach; Leudtke; Unsworth; Boundy; Nowak; Scripko; Elder; Jackson; Hoffman; Evora; Rao; Molinoff; Childers; Ehrenkaufer Journal of Medicinal Chemistry, 1993 , vol. 36, # 23 p. 3707 - 3720]

Synthesis and Structure-Activity Relationships of N-(1-Benzy...

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