Orexin receptor antagonist 4
Modify Date: 2024-01-11 22:15:31
Orexin receptor antagonist 4 structure
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Common Name | Orexin receptor antagonist 4 | ||
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| CAS Number | 2251017-69-1 | Molecular Weight | 408.47 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C23H25FN4O2 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Orexin receptor antagonist 4Orexin receptor antagonist 4 is potent and selective orexin 2 receptor (OX2R) antagonist with an IC50 of 4.27 nM. Orexin receptor antagonist 4 is 61-fold selective for the OX2R over the OX1R (IC50 of 295 nM) (WO2018206959A1; example 1)[1]. |
| Name | Orexin receptor antagonist 4 |
|---|
| Description | Orexin receptor antagonist 4 is potent and selective orexin 2 receptor (OX2R) antagonist with an IC50 of 4.27 nM. Orexin receptor antagonist 4 is 61-fold selective for the OX2R over the OX1R (IC50 of 295 nM) (WO2018206959A1; example 1)[1]. |
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| Related Catalog | |
| Target |
OX2 Receptor:4.27 nM (IC50) OX1 Receptor:295 nM (IC50) |
| References |
[1]. David Sheppard, et al. Orexin receptor antagonists. WO2018206959A1 |
| Molecular Formula | C23H25FN4O2 |
|---|---|
| Molecular Weight | 408.47 |