PG 106 TFA

Modify Date: 2024-01-11 08:18:05

PG 106 TFA structure	Common Name	PG 106 TFA
	CAS Number	944111-22-2	Molecular Weight	1008.18000
	Density	1.40±0.1 g/cm3 (20 °C, 760 mmHg)	Boiling Point	N/A
	Molecular Formula	C₅₁H₆₉N₁₃O₉	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of PG 106 TFA

PG106 is a potent and selective human melanocortin 3 (hMC3) receptor antagonist (IC50=210 nM) and has noactivity at hMC4 receptors (EC50=9900 nM) and hMC5 receptor[1].

Name	L-Lysinamide, N-acetyl-L-norleucyl-L-α-aspartyl-β-alanyl-3-(2-naphthalenyl)-D-alanyl-L-arginyl-L-tryptophyl-, (2→7)-lactam
Synonym	More Synonyms

Description	PG106 is a potent and selective human melanocortin 3 (hMC3) receptor antagonist (IC50=210 nM) and has noactivity at hMC4 receptors (EC50=9900 nM) and hMC5 receptor[1].
Related Catalog	Research Areas >> Inflammation/Immunology Signaling Pathways >> GPCR/G Protein >> Melanocortin Receptor
Target	IC50: 210 nM (hMC3 receptor) EC50: 9900 nM (hMC4 receptor)[1]
References	[1]. Paolo Grieco, et al. Further structure-activity studies of lactam derivatives of MT-II and SHU-9119: their activity and selectivity at human melanocortin receptors 3, 4, and 5. Peptides

Density	1.40±0.1 g/cm3 (20 °C, 760 mmHg)
Molecular Formula	C₅₁H₆₉N₁₃O₉
Molecular Weight	1008.18000
Exact Mass	1007.53000
PSA	353.58000
LogP	4.81610

MMPIP hydrochloride

DC Chemicals Limited
China
Product Name: PG106
Price: $Inquiry/250mg $Inquiry/100mg $Inquiry/1g
Purity: 98.0%
Stocking Period: 3 Day
Contact: Tony Cao

Zhejiang Hangyu API Co., Ltd
China
Product Name: PG106
Price: $Inquiry/1kg
Purity: 99.0%
Stocking Period: 1 Day
Contact: Vinnie

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