Gsk466317a

Modify Date: 2025-09-11 10:18:35

Gsk466317a structure	Common Name	Gsk466317a
	CAS Number	864082-48-4	Molecular Weight	448.83
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₁H₁₆ClF₃N₄O₂	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of Gsk466317a

GSK466317A is a PKA inhibitor, with an IC50 of 12.59 μM. GSK466317A also inhibits GRK1, GRK2, and GRK5, with IC50s of 1000, 31.62, and 39.81 μM, respectively[1].

Name	GSK466317A

Description	GSK466317A is a PKA inhibitor, with an IC50 of 12.59 μM. GSK466317A also inhibits GRK1, GRK2, and GRK5, with IC50s of 1000, 31.62, and 39.81 μM, respectively[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Protein Tyrosine Kinase/RTK >> PKA Signaling Pathways >> Stem Cell/Wnt >> PKA Research Areas >> Neurological Disease
Target	PKA:12.59 μM (IC50)
References	[1]. Homan KT, et, al. Identification and structure-function analysis of subfamily selective G protein-coupled receptor kinase inhibitors. ACS Chem Biol. 2015 Jan 16;10(1):310-9.

Molecular Formula	C₂₁H₁₆ClF₃N₄O₂
Molecular Weight	448.83
InChIKey	OYNBTBJATZVIGH-UHFFFAOYSA-N
SMILES	CC1=C(C(=O)Nc2cc(Cl)c3[nH]ncc3c2)C(c2ccc(C(F)(F)F)cc2)CC(=O)N1

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.

Shanghai Nianxing Industrial Co., Ltd
China
Product Name: Gsk466317a
Price: Check
Purity: 98.0%
Delivery: 10 Day
Contact: Yang
Email: sales@echemcloud.com

DC Chemicals Limited
China
Product Name: Gsk466317a
Price: ￥Inquiry/100mg ￥Inquiry/250mg ￥Inquiry/1g
Purity: 98.0%
Delivery: 10 Day
Contact: Tony Cao
Email: sales@dcchemicals.com

Get all suppliers and price by the below link:

Gsk466317a suppliers

Gsk466317a price