H4 Receptor antagonist 1

Modify Date: 2024-01-02 18:32:38

H4 Receptor antagonist 1 structure	Common Name	H4 Receptor antagonist 1
	CAS Number	848217-00-5	Molecular Weight	316.79
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₁₆H₁₇ClN₄O	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of H4 Receptor antagonist 1

H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.

Name	H4 Receptor antagonist 1

Description	H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Histamine Receptor Signaling Pathways >> Immunology/Inflammation >> Histamine Receptor Research Areas >> Neurological Disease
Target	H4 receptor:19 nM (IC50)
In Vitro	H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM[1].
In Vivo	H4 Receptor antagonist 1 indicates that metabolic stability in rat microsomes is very low with only 1% parent compound remaining after 10 min incubation[1].
References	[1]. Cramp S, et al. Identification and hit-to-lead exploration of a novel series of histamine H4 receptor inverse agonists. Bioorg Med Chem Lett. 2010 Apr 15;20(8):2516-9.

Molecular Formula	C₁₆H₁₇ClN₄O
Molecular Weight	316.79
Storage condition	2-8℃

DC Chemicals Limited
China
Product Name: H4 Receptor antagonist 1
Price: $Inquiry/100mg $Inquiry/250mg $Inquiry/1g
Purity: 98.0%
Stocking Period: 3 Day
Contact: Tony Cao

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Price: ￥990/10 mM * 1 mL in DMSO

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