Name | H4 Receptor antagonist 1 |
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Description | H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. |
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Related Catalog | |
Target |
H4 receptor:19 nM (IC50) |
In Vitro | H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM[1]. |
In Vivo | H4 Receptor antagonist 1 indicates that metabolic stability in rat microsomes is very low with only 1% parent compound remaining after 10 min incubation[1]. |
References |
Molecular Formula | C16H17ClN4O |
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Molecular Weight | 316.79 |
Storage condition | 2-8℃ |