Dynorphin A trifluoroacetate salt
Dynorphin A trifluoroacetate salt structure
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Common Name | Dynorphin A trifluoroacetate salt | ||
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| CAS Number | 80448-90-4 | Molecular Weight | 2147.484 | |
| Density | 1.5±0.1 g/cm3 | Boiling Point | N/A | |
| Molecular Formula | C99H155N31O23 | Melting Point | N/A | |
| MSDS | Chinese USA | Flash Point | N/A | |
Use of Dynorphin A trifluoroacetate saltDynorphin A, an endogenous opioid peptide, is a highy potent kappa opioid receptor (KOR) activator. Dynorphin A also serve as an agonist for other opioid receptors, such as mu (MOR) and delta (DOR)[1]. |
| Name | Dynorphin A |
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| Synonym | More Synonyms |
| Description | Dynorphin A, an endogenous opioid peptide, is a highy potent kappa opioid receptor (KOR) activator. Dynorphin A also serve as an agonist for other opioid receptors, such as mu (MOR) and delta (DOR)[1]. |
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| Related Catalog | |
| References |
| Density | 1.5±0.1 g/cm3 |
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| Molecular Formula | C99H155N31O23 |
| Molecular Weight | 2147.484 |
| Exact Mass | 2146.191162 |
| PSA | 917.37000 |
| LogP | -1.52 |
| Index of Refraction | 1.669 |
| Storage condition | −20°C |
| Personal Protective Equipment | Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter |
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| Safety Phrases | 22-24/25 |
| RIDADR | NONH for all modes of transport |
| WGK Germany | 3 |
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Dynorphin A as a potential endogenous ligand for four members of the opioid receptor gene family.
J. Pharmacol. Exp. Ther. 286 , 136-141, (1998) Dynorphin A is an endogenous opioid peptide that activates the kappa opioid receptor (KOR) with high potency. Some studies also showed that the distribution and functional activity of dynorphin A are ... |
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Structure-activity relationship studies of dynorphin A and related peptides.
Peptides 19 , 1277-1292, (1998) An up-to-date review is presented covering all the available information concerning the isolation, discovery, synthesis, conformation, receptor binding characteristics, pharmacological properties and ... |
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The kappa opioid receptor and dynorphin co-localize in vasopressin magnocellular neurosecretory neurons in guinea-pig hypothalamus.
Neuroscience 96 , 373-383, (2000) The relationship between the cloned kappa opioid receptor, dynorphin, and the neurohypophysial hormones vasopressin and oxytocin was analysed in the guinea-pig hypothalamic magnocellular neurosecretor... |
| Dynorphin acetate |
| DYNORPHIN A PORCINE |
| L-Tyrosylglycylglycyl-L-phenylalanyl-L-leucyl-L-arginyl-L-arginyl-L-isoleucyl-L-arginyl-L-prolyl-L-lysyl-L-leucyl-L-lysyl-L-tryptophyl-L-α-aspartyl-L-asparaginyl-L-glutamine |
| YGGFLRRIRPKLKWDNQ |
| L-Glutamine, L-tyrosylglycylglycyl-L-phenylalanyl-L-leucyl-L-arginyl-L-arginyl-L-isoleucyl-L-arginyl-L-prolyl-L-lysyl-L-leucyl-L-lysyl-L-tryptophyl-L-α-aspartyl-L-asparaginyl- |
| DYNORPHIN A AMIDE |