Firazorexton hydrate
Modify Date: 2024-01-13 06:06:04
Firazorexton hydrate structure
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Common Name | Firazorexton hydrate | ||
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| CAS Number | 2861934-86-1 | Molecular Weight | 497.53 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C22H25F3N2O4S.3/2H2O | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Firazorexton hydrateFirazorexton hydrate (TAK-994) is a potent, brain-penetrant, and orally active orexin type 2 receptor (OX2R) agonist (EC50: 19 nM). Firazorexton hydrate inhibits fragmentation of wakefulness and cataplexy-like episodes in mouse models of narcolepsy[1]. |
| Name | Firazorexton hydrate |
|---|
| Description | Firazorexton hydrate (TAK-994) is a potent, brain-penetrant, and orally active orexin type 2 receptor (OX2R) agonist (EC50: 19 nM). Firazorexton hydrate inhibits fragmentation of wakefulness and cataplexy-like episodes in mouse models of narcolepsy[1]. |
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| Related Catalog | |
| Target |
EC50: 19 nM (OX2R)[1] |
| References |
| Molecular Formula | C22H25F3N2O4S.3/2H2O |
|---|---|
| Molecular Weight | 497.53 |