BRD4-BD1-IN-2

Modify Date: 2024-04-02 19:45:02

BRD4-BD1-IN-2 structure	Common Name	BRD4-BD1-IN-2
	CAS Number	2761321-26-8	Molecular Weight	583.07
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₀H₁₅Br₃N₄O₂	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of BRD4-BD1-IN-2

BRD4-BD1-IN-2 is a selective BRD4-BD1 inhibitor, with an IC50 of 2.51 µM (20-times greater than that of BD2). BRD4-BD1-IN-2 can be used in studies of cancer and cardiovascular diseases[1].

Name	BRD4-BD1-IN-2

Description	BRD4-BD1-IN-2 is a selective BRD4-BD1 inhibitor, with an IC50 of 2.51 µM (20-times greater than that of BD2). BRD4-BD1-IN-2 can be used in studies of cancer and cardiovascular diseases[1].
Related Catalog	Research Areas >> Cancer Research Areas >> Cardiovascular Disease Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain
Target	BRD4-BD1:2.51 μM (IC50) BRD4-BD2:＞50 μM (IC50)
References	[1]. Chang Y, et al. Design, synthesis, biological evaluation, and molecular docking of 1, 7-dibenzyl-substituted theophylline derivatives as novel BRD4-BD1-selective inhibitors. Medicinal Chemistry Research, 2021, 30(8): 1453-1468.

Molecular Formula	C₂₀H₁₅Br₃N₄O₂
Molecular Weight	583.07