PROTAC FAK degrader 1

Modify Date: 2025-09-18 15:39:12

PROTAC FAK degrader 1 Structure
PROTAC FAK degrader 1 structure
Common Name PROTAC FAK degrader 1
CAS Number 2301916-69-6 Molecular Weight 996.13
Density N/A Boiling Point N/A
Molecular Formula C47H56F3N9O8S2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of PROTAC FAK degrader 1


PROTAC FAK degrader 1 is a selective and potent focal adhesion kinase (Fak) degrader with an IC50 of 6.5 nM, DC50 of 3 nM[1].

 Names

Name PROTAC FAK degrader 1

 PROTAC FAK degrader 1 Biological Activity

Description PROTAC FAK degrader 1 is a selective and potent focal adhesion kinase (Fak) degrader with an IC50 of 6.5 nM, DC50 of 3 nM[1].
Related Catalog
Target

IC50: 6.5 nM (Focal adhesion kinase) DC50: 3 nM (Focal adhesion kinase)[1]

References

[1]. Cromm PM, et al. Addressing Kinase-Independent Functions of Fak via PROTAC-Mediated Degradation. J Am Chem Soc. 2018 Dec 12;140(49):17019-17026.

 Chemical & Physical Properties

Molecular Formula C47H56F3N9O8S2
Molecular Weight 996.13
Storage condition -20°C
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