PROTAC BET Degrader-1

Modify Date: 2025-08-24 18:10:12

PROTAC BET Degrader-1 structure	Common Name	PROTAC BET Degrader-1
	CAS Number	2093386-22-0	Molecular Weight	871.9
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₄₄H₄₅N₁₁O₉	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of PROTAC BET Degrader-1

PROTAC BET Degrader-1 is a potent BET degrader based on PROTAC, decreasing BRD2, BRD3, and BRD4 protein levels at low concentration.

Name	PROTAC 11

Description	PROTAC BET Degrader-1 is a potent BET degrader based on PROTAC, decreasing BRD2, BRD3, and BRD4 protein levels at low concentration.
Related Catalog	Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain Signaling Pathways >> PROTAC >> PROTAC Research Areas >> Cancer
Target	BET[1]
In Vitro	PROTAC BET Degrader-1 (Compound 9) is a potent BET degrader based on PROTAC, decreases the level of BRD2, BRD3, and BRD4 proteins in RS4;11 cells at 3-10 nM, and inhibits the growth of this cell line with an IC50 of 4.3 nM, and 45.5 nM for MOLM-13 cells[1].
References	[1]. Zhou B, et al. Discovery of a Small-Molecule Degrader of Bromodomain and Extra-Terminal (BET) Proteins with Picomolar Cellular Potencies and Capable of Achieving Tumor Regression. J Med Chem. 2018 Jan 25;61(2):462-481.

Molecular Formula	C₄₄H₄₅N₁₁O₉
Molecular Weight	871.9

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Shanghai Nianxing Industrial Co., Ltd
China
Product Name: PROTAC BET Degrader-1
Price: Check
Purity: 98.0%
Delivery: 10 Day
Contact: Yang
Email: sales@echemcloud.com

DC Chemicals Limited
China
Product Name: PROTAC BET Degrader-1
Price: $Inquiry/1g
Purity: 98.0%
Delivery: 1 Day
Contact: Tony Cao
Email: sales@dcchemicals.com

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PROTAC BET Degrader-1 suppliers

Price: ￥8152/10 mM * 1 mL in DMSO

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