CBP/p300-IN-10
Modify Date: 2025-11-25 00:51:31
CBP/p300-IN-10 structure
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Common Name | CBP/p300-IN-10 | ||
|---|---|---|---|---|
| CAS Number | 2259641-71-7 | Molecular Weight | 537.48 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C25H24F5N5O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of CBP/p300-IN-10CBP/p300-IN-10 is a highly potent histone acetyltransferase EP300 and CREBBP with IC50 values of 26 nM and 39 nM, respectively. CBP/p300-IN-10 can be used to research anticancer[1]. |
| Name | CBP/p300-IN-10 |
|---|
| Description | CBP/p300-IN-10 is a highly potent histone acetyltransferase EP300 and CREBBP with IC50 values of 26 nM and 39 nM, respectively. CBP/p300-IN-10 can be used to research anticancer[1]. |
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| Related Catalog | |
| Target |
EP300:26 nM (IC50) CREBBP:39 nM (IC50) |
| In Vitro | CBP/p300-IN-10 (example 84) (0-1 μM; 3 h) inhibit H3K27Ac activity in LK2 cells with an IC50 of 22 nM[1]. CBP/p300-IN-10 (38 nM-10 mM; 3 days) has inhibitory activity against LK2 and TE-8[1]. Cell Proliferation Assay[1] Cell Line: LK2 and TE-8 Concentration: 38 nM-10 mM Incubation Time: 3 days Result: Inhibited LK2 and TE-8 with GI50s of 97.163 nM and 152.484 nM, respectively. |
| References |
| Molecular Formula | C25H24F5N5O3 |
|---|---|
| Molecular Weight | 537.48 |