CBP/p300-IN-17

Modify Date: 2025-08-28 22:28:28

CBP/p300-IN-17 Structure
CBP/p300-IN-17 structure
 Common Name CBP/p300-IN-17
CAS Number 2259640-87-2 Molecular Weight 432.51
Density N/A Boiling Point N/A
Molecular Formula C25H28N4O3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of CBP/p300-IN-17


CBP/p300-IN-17 (compound 7) is a potent EP300/CBP HAT inhibitor with IC50s of 0.18, 0.69 µM for HAT EP300 and LK2 H3K27, respectively[1].

 Names

Name CBP/p300-IN-17

 CBP/p300-IN-17 Biological Activity

Description CBP/p300-IN-17 (compound 7) is a potent EP300/CBP HAT inhibitor with IC50s of 0.18, 0.69 µM for HAT EP300 and LK2 H3K27, respectively[1].
Related Catalog
Target

EP300:0.18 μM (IC50)

LK2 H3K27:0.69 μM (IC50)

References

[1]. Kanada R, et al. Discovery of EP300/CBP histone acetyltransferase inhibitors through scaffold hopping of 1,4-oxazepane ring. Bioorg Med Chem Lett. 2022 Jun 15;66:128726.

 Chemical & Physical Properties

Molecular Formula C25H28N4O3
Molecular Weight 432.51
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Chemsrc provides CBP/p300-IN-17(CAS#:2259640-87-2) MSDS, density, melting point, boiling point, structure, formula, molecular weight etc. Articles of CBP/p300-IN-17 are included as well.>> amp version: CBP/p300-IN-17

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