APJ receptor agonist 7
Modify Date: 2024-01-14 10:55:39
APJ receptor agonist 7 structure
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Common Name | APJ receptor agonist 7 | ||
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| CAS Number | 2100850-28-8 | Molecular Weight | 550.73 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C32H46N4O4 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of APJ receptor agonist 7APJ receptor agonist 7 (compound 37) is a potent and orally active APJ (apelin receptor) agonist, with Ki of 0.059 μM. APJ receptor agonist 7 has EC50 values of 0.070 , 0.097, and 0.063 μM for calcium, cAMP, and β-arrestin, respectively[1]. |
| Name | APJ receptor agonist 7 |
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| Description | APJ receptor agonist 7 (compound 37) is a potent and orally active APJ (apelin receptor) agonist, with Ki of 0.059 μM. APJ receptor agonist 7 has EC50 values of 0.070 , 0.097, and 0.063 μM for calcium, cAMP, and β-arrestin, respectively[1]. |
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| Related Catalog | |
| Target |
EC50: 0.063 ± 0.004 μM (Apelin Receptor β-arrestin), 0.070 ± 0.009 μM (Apelin Receptor calcium), 0.097 ± 0.032 μM (Apelin Receptor cAMP), >10 μM (AT1 calcium)[1] |
| References |
| Molecular Formula | C32H46N4O4 |
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| Molecular Weight | 550.73 |