dBET23

Modify Date: 2024-04-06 23:24:48

dBET23 Structure
dBET23 structure
Common Name dBET23
CAS Number 1957234-83-1 Molecular Weight 885.39
Density N/A Boiling Point N/A
Molecular Formula C43H45ClN8O9S Melting Point N/A
MSDS N/A Flash Point N/A

 Use of dBET23


dBET23 is a BRD4 heterobifunctional small-molecule ligand (PROTAC), exhibits significant and selective degradation of BRD4 BD1 (DC50/5h=50 nM) in cellular degradation assays.

 Names

Name dBET23

 dBET23 Biological Activity

Description dBET23 is a BRD4 heterobifunctional small-molecule ligand (PROTAC), exhibits significant and selective degradation of BRD4 BD1 (DC50/5h=50 nM) in cellular degradation assays.
References References 1. Nowak RP, et al. Nat Chem Biol. 2018 Jun 11. doi: 10.1038/s41589-018-0055-y. View Related Products by Target PROTAC

 Chemical & Physical Properties

Molecular Formula C43H45ClN8O9S
Molecular Weight 885.39

 Safety Information

Hazard Codes Xi