Name | dBET23 |
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Description | dBET23 is a BRD4 heterobifunctional small-molecule ligand (PROTAC), exhibits significant and selective degradation of BRD4 BD1 (DC50/5h=50 nM) in cellular degradation assays. |
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References | References 1. Nowak RP, et al. Nat Chem Biol. 2018 Jun 11. doi: 10.1038/s41589-018-0055-y. View Related Products by Target PROTAC |
Molecular Formula | C43H45ClN8O9S |
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Molecular Weight | 885.39 |
Hazard Codes | Xi |
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