PW0464
Modify Date: 2024-01-08 12:25:45
PW0464 structure
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Common Name | PW0464 | ||
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| CAS Number | 1643462-93-4 | Molecular Weight | 389.35 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C19H17F2N3O4 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of PW0464PW0464, a nanomolar potent complete G protein biased ligand, is a noncatechol D1R agonist, with an EC50 of 5.8 nM (Gs-cAMP)[1]. |
| Name | PW0464 |
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| Description | PW0464, a nanomolar potent complete G protein biased ligand, is a noncatechol D1R agonist, with an EC50 of 5.8 nM (Gs-cAMP)[1]. |
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| Related Catalog | |
| In Vitro | PW0464 (compound 24) is found to elicit complete G protein bias, showing no activity for D1R-mediated β-arrestin recruitment[1]. PW0464 (compound 24), the non-catechol agonist, forms bonds with S1985.42 and S2025.46 via its fluorine atom[2]. |
| References |
| Molecular Formula | C19H17F2N3O4 |
|---|---|
| Molecular Weight | 389.35 |