(Des-Arg9)-Bradykinin acetate salt structure
|
Common Name | (Des-Arg9)-Bradykinin acetate salt | ||
|---|---|---|---|---|
| CAS Number | 15958-92-6 | Molecular Weight | 904.023 | |
| Density | 1.5±0.1 g/cm3 | Boiling Point | N/A | |
| Molecular Formula | C44H61N11O10 | Melting Point | N/A | |
| MSDS | USA | Flash Point | N/A | |
Use of (Des-Arg9)-Bradykinin acetate salt[Des-Arg9]-Bradykinin is a Bradykinin (B1) receptor agonist that displays selectivity for B1 over B2 receptors. |
| Name | [Des-Arg9]-Bradykinin |
|---|---|
| Synonym | More Synonyms |
| Description | [Des-Arg9]-Bradykinin is a Bradykinin (B1) receptor agonist that displays selectivity for B1 over B2 receptors. |
|---|---|
| Related Catalog | |
| Target |
Bradykinin (B1) receptor[1] |
| In Vitro | The B2 receptor mediates the action of bradykinin (BK) and lysyl-bradykinin (Lys-BK), the first set of bioactive kinins formed in response to injury from kininogen precursors through the actions of plasma and tissue kallikreins, whereas the B1 receptor mediates the action of [Des-Arg9]-Bradykinin (des-Arg9-BK) and Lys-des-Arg Arg9-BK, the second set of bioactive kinins formed through the actions of carboxypeptidases on BK and Lys-BK, respectively[1]. |
| References |
| Density | 1.5±0.1 g/cm3 |
|---|---|
| Molecular Formula | C44H61N11O10 |
| Molecular Weight | 904.023 |
| Exact Mass | 903.460266 |
| PSA | 322.78000 |
| LogP | 0.64 |
| Index of Refraction | 1.687 |
| Storage condition | -20°C |
|
~%
(Des-Arg9)-Brad... CAS#:15958-92-6 |
| Literature: Umetsu, H.; Ichishima, E. Phytochemistry (Elsevier), 1983 , vol. 22, # 2 p. 591 - 592 |
| Precursor 1 | |
|---|---|
| DownStream 0 | |
| L-phenylalanine, N-[[(2S)-1-[(2S)-2-[[(1Z,2S)-2-[[(1E)-2-[[(1Z)-[(2S)-1-[[(2S)-1-[(2S)-2-amino-5-[(aminoiminomethyl)amino]-1-oxopentyl]-2-pyrrolidinyl]carbonyl]-2-pyrrolidinyl]hydroxymethylene]amino]-1-hydroxyethylidene]amino]-1-hydroxy-3-phenylpropylidene]amino]-3-hydroxy-1-oxopropyl]-2-pyrrolidinyl]hydroxymethylene]-, (Z)- |
| 1-8-Bradykinin |
| des-arginine9-bradykinin |
| bradykinin fragment 1-8 |
| 9-Des-Arg-bk |
| [des-Arg(9)]-bradykinin |
| 9-De-Arg-bradykinin |
| L-Phenylalanine, N-(diaminomethylene)-L-ornithyl-L-prolyl-L-prolylglycyl-L-phenylalanyl-L-seryl-L-prolyl- |
| des-Arg9-bradykinin |
| RPPGFSPF |
| DABK |
| N-(Diaminomethylene)-L-ornithyl-L-prolyl-L-prolylglycyl-L-phenylalanyl-L-seryl-L-prolyl-L-phenylalanine |
| des-Arg9-BK |
| Bradykinin[Des-Arg9] |