GPR4 antagonist 3

Modify Date: 2024-01-14 15:13:26

GPR4 antagonist 3 structure	Common Name	GPR4 antagonist 3
	CAS Number	1401728-56-0	Molecular Weight	416.52
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₄H₂₈N₆O	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of GPR4 antagonist 3

GPR4 antagonist 3 is a selective, and orally available GPR4 antagonist with an IC50 of 70 nM[1]. Anti-inflammatory activities[1].

Name	GPR4 antagonist 3

Description	GPR4 antagonist 3 is a selective, and orally available GPR4 antagonist with an IC50 of 70 nM[1]. Anti-inflammatory activities[1].
Related Catalog	Signaling Pathways >> Others >> Others Research Areas >> Inflammation/Immunology
Target	IC50: 70 nM (GPR4)[1].
In Vivo	GPR4 antagonist 3 shows a significant anti-inflammatory effect in the rat antigen induced arthritis model after oral administration at 30 mg/kg bid[1].GPR4 antagonist 3 also prevents angiogenesis in the mouse chamber model as well as pain as demonstrated in the rat complete Freund’s adjuvant model[1].
References	[1]. Velcicky J, et al. Development of Selective, Orally Active GPR4 Antagonists with Modulatory Effects on Nociception, Inflammation, and Angiogenesis. J Med Chem. 2017 May 11;60(9):3672-3683.

Molecular Formula	C₂₄H₂₈N₆O
Molecular Weight	416.52

DC Chemicals Limited
China
Product Name: GPR4 antagonist 3
Price: $800.0/100mg $1500.0/250mg $3000.0/1g
Purity: 98.0%
Stocking Period: 3 Day
Contact: Tony Cao

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