glucagon receptor antagonists-4

Modify Date: 2025-08-21 10:24:37

glucagon receptor antagonists-4 structure	Common Name	glucagon receptor antagonists-4
	CAS Number	1393124-08-7	Molecular Weight	503.513
	Density	1.3±0.1 g/cm3	Boiling Point	675.0±55.0 °C at 760 mmHg
	Molecular Formula	C₂₆H₂₈F₃N₃O₄	Melting Point	N/A
	MSDS	N/A	Flash Point	362.0±31.5 °C

Use of glucagon receptor antagonists-4

Glucagon receptor antagonists-4 is a highly potent glucagon receptor antagonist. It displays low in vivo clearance and excellent oral bioavailability in both rats and dogs.

Name	N-{4-[(1S)-1-{3,5-Dimethyl-4-[4-(trifluoromethyl)-1H-pyrazol-1-yl]phenoxy}butyl]benzoyl}-β-alanine
Synonym	More Synonyms

Description	Glucagon receptor antagonists-4 is a highly potent glucagon receptor antagonist. It displays low in vivo clearance and excellent oral bioavailability in both rats and dogs.
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Glucagon Receptor Research Areas >> Metabolic Disease
References	[1]. Guzman-Perez A et al. The design and synthesis of a potent glucagon receptor antagonist with favorable physicochemical andpharmacokinetic properties as a candidate for the treatment of type 2 diabetes mellitus. Bioorg Med Chem Lett, 2013 May 15, 23(10):3051-8. [2]. Esther C.Y. Lee et al. Identification of a novel conformationally constrained glucagon receptor antagonist. Bioorg Med Chem Lett, 2014 Feb 1, 24(3):839-44.

Description

Glucagon receptor antagonists-4 is a highly potent glucagon receptor antagonist. It displays low in vivo clearance and excellent oral bioavailability in both rats and dogs.

Related Catalog

Signaling Pathways >> GPCR/G Protein >> Glucagon Receptor

Research Areas >> Metabolic Disease

References

[1]. Guzman-Perez A et al. The design and synthesis of a potent glucagon receptor antagonist with favorable physicochemical andpharmacokinetic properties as a candidate for the treatment of type 2 diabetes mellitus. Bioorg Med Chem Lett, 2013 May 15, 23(10):3051-8.

[2]. Esther C.Y. Lee et al. Identification of a novel conformationally constrained glucagon receptor antagonist. Bioorg Med Chem Lett, 2014 Feb 1, 24(3):839-44.

Density	1.3±0.1 g/cm3
Boiling Point	675.0±55.0 °C at 760 mmHg
Molecular Formula	C₂₆H₂₈F₃N₃O₄
Molecular Weight	503.513
Flash Point	362.0±31.5 °C
Exact Mass	503.203186
LogP	5.44
Vapour Pressure	0.0±2.2 mmHg at 25°C
Index of Refraction	1.563

N-{4-[(1S)-1-{3,5-Dimethyl-4-[4-(trifluoromethyl)-1H-pyrazol-1-yl]phenoxy}butyl]benzoyl}-β-alanine

β-Alanine, N-[4-[(1S)-1-[3,5-dimethyl-4-[4-(trifluoromethyl)-1H-pyrazol-1-yl]phenoxy]butyl]benzoyl]-

glucagon receptor antagonists-4

PF-06291874

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China
Product Name: glucagon receptor antagonists-4
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Price: $465/10mM*1mLinDMSO

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glucagon receptor antagonists-4

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