CCK-A receptor inhibitor 1

Modify Date: 2024-01-11 23:22:09

CCK-A receptor inhibitor 1 structure	Common Name	CCK-A receptor inhibitor 1
	CAS Number	137004-80-9	Molecular Weight	477.61
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₅H₃₅NO₆S	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of CCK-A receptor inhibitor 1

CCK-A receptor inhibitor 1 is a cholecystokinin A (CCK-A) receptor inhibitor with a binging IC50 of 340 nM.

Name	CCK-A receptor inhibitor 1

Description	CCK-A receptor inhibitor 1 is a cholecystokinin A (CCK-A) receptor inhibitor with a binging IC50 of 340 nM.
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Cholecystokinin Receptor Research Areas >> Metabolic Disease
Target	IC50: 340 nM (CCK-A receptor)[1]
In Vitro	CCK-A receptor inhibitor 1 (Compound 7c) is a naphthyl sulfone derivative, which is synthesized and tested for cholecystokinin A (CCK-A) receptor inhibitory activity in order to study structure-activity relationships. Significant CCK-A receptor inhibitory activities are found in CCK-A receptor inhibitor 1 having very hydrophobic sidechains[1].
References	[1]. Ajisawa Y, et al. [Studies on the synthesis of cholecystokinin A receptor antagonists. III. Synthesis and cholecystokinin A receptor inhibitory activities of naphthyl sulfone derivatives]. Yakugaku Zasshi. 1996 Aug;116(8):647-56.

Molecular Formula	C₂₅H₃₅NO₆S
Molecular Weight	477.61