threo Ifenprodil hemitartrate structure
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Common Name | threo Ifenprodil hemitartrate | ||
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CAS Number | 1312991-83-5 | Molecular Weight | 400.50 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C21H27NO2.1/2C4H6O6 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of threo Ifenprodil hemitartratethreo Ifenprodil hemitartrate is a σ receptor agonist, with Kis of 59.1 and 2 nM for σ1 and σ2 receptors, respectively. threo Ifenprodil hemitartrate is also a NR2B subunit-selective NMDA receptor antagonist (IC50=0.22 μM). threo Ifenprodil hemitartrate is a hERG potassium channel inhibitor, with an IC 50 of 88 nM, showing antiarrhythmic activity[1][2][3]. |
Name | threo Ifenprodil hemitartrate |
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Description | threo Ifenprodil hemitartrate is a σ receptor agonist, with Kis of 59.1 and 2 nM for σ1 and σ2 receptors, respectively. threo Ifenprodil hemitartrate is also a NR2B subunit-selective NMDA receptor antagonist (IC50=0.22 μM). threo Ifenprodil hemitartrate is a hERG potassium channel inhibitor, with an IC 50 of 88 nM, showing antiarrhythmic activity[1][2][3]. |
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Related Catalog | |
Target |
IC50: 0.22 μM (NMDA)[1]. |
References |
Molecular Formula | C21H27NO2.1/2C4H6O6 |
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Molecular Weight | 400.50 |
Exact Mass | 1600.849609 |