[D-Ala2] -Deltorphin II structure
|
Common Name | [D-Ala2] -Deltorphin II | ||
|---|---|---|---|---|
| CAS Number | 122752-16-3 | Molecular Weight | 782.88300 | |
| Density | 1.272 g/cm3 | Boiling Point | 1256.2ºC at 760 mmHg | |
| Molecular Formula | C38H54N8O10 | Melting Point | N/A | |
| MSDS | Chinese USA | Flash Point | 713.5ºC | |
Use of [D-Ala2] -Deltorphin IIDeltorphin 2 is a selective peptide agonit for the δ opioid receptor. |
| Name | [D-Ala2]-Deltorphin II |
|---|---|
| Synonym | More Synonyms |
| Description | Deltorphin 2 is a selective peptide agonit for the δ opioid receptor. |
|---|---|
| Related Catalog | |
| Target |
δ opioid receptor[1] |
| In Vitro | Deltorphin 2 ([D-Ala2]-Deltorphin II) is enzymatically stable, amphibian heptapeptides that has a high affinity and selectivity for delta-opioid receptor. Deltorphin 2 is the most selective natural delta opioid receptor agonist[1]. |
| References |
| Density | 1.272 g/cm3 |
|---|---|
| Boiling Point | 1256.2ºC at 760 mmHg |
| Molecular Formula | C38H54N8O10 |
| Molecular Weight | 782.88300 |
| Flash Point | 713.5ºC |
| Exact Mass | 782.39600 |
| PSA | 301.24000 |
| LogP | 2.47290 |
| Vapour Pressure | 0mmHg at 25°C |
| Index of Refraction | 1.575 |
| Storage condition | -20°C |
| Personal Protective Equipment | Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter |
|---|---|
| RIDADR | NONH for all modes of transport |
|
Membrane partitioning of various delta-opioid receptor forms before and after agonist activations: the effect of cholesterol.
Biochim. Biophys. Acta 1778(6) , 1483-92, (2008) Lipid rafts depicted as densely packed and thicker membrane microdomains, based on the dynamic clustering of cholesterol and sphingolipids, may help as platforms involved in a wide variety of cellular... |
|
|
Delta opioid receptor-mediated analgesia is not altered in preprotachykinin A knockout mice.
Eur. J. Neurosci. 32(11) , 1921-9, (2010) We have shown that delta opioid receptor (DOPR)-mediated analgesia was enhanced in the complete Freund's adjuvant (CFA) model of inflammation. This effect is thought to originate from translocation of... |
|
|
Functional identification of a novel transport system for endogenous and synthetic opioid peptides in the rabbit conjunctival epithelial cell line CJVE.
Pharm. Res. 26(5) , 1226-35, (2009) To investigate whether conjunctival epithelial cells express transport processes for opioid peptides.We monitored the uptake of [(3)H]deltorphin II and [(3)H]DADLE, two hydrolysis-resistant synthetic ... |
| Tyr-D-Ala-Phe-Glu-Val-Val-Gly amide |
| M.W. 782.89 C38H54N8O10 |
| DELTORPHIN B |
| DADELT II |
| H-Tyr-D-Ala-Phe-Glu-Val-Val-Gly-NH2 |
| H2N-Tyr-D-Ala-Phe-Glu-Val-Val-Gly-NH2 |
| deltorphin II |
| TYR-D-ALA-PHE-GLU-VAL-VAL-GLY-NH2 |
| DELTORPHIN II |
| Deltorphin 2 |