3-Hydroxy agomelatine D3

Modify Date: 2024-01-30 06:57:10

3-Hydroxy agomelatine D3 Structure
3-Hydroxy agomelatine D3 structure
Common Name 3-Hydroxy agomelatine D3
CAS Number 1079774-23-4 Molecular Weight 262.32
Density N/A Boiling Point N/A
Molecular Formula C15H14D3NO3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of 3-Hydroxy agomelatine D3


3-Hydroxy agomelatine D3 is a deuterium labeled 3-Hydroxy agomelatine. 3-Hydroxy agomelatine is a 5-HT2C receptor antagonist with an IC50 of 3.2 μM and a Ki of 1.8 μM[1].

 Names

Name 3-Hydroxy agomelatine D3

 3-Hydroxy agomelatine D3 Biological Activity

Description 3-Hydroxy agomelatine D3 is a deuterium labeled 3-Hydroxy agomelatine. 3-Hydroxy agomelatine is a 5-HT2C receptor antagonist with an IC50 of 3.2 μM and a Ki of 1.8 μM[1].
Related Catalog
Target

5-HT2C Receptor:3.2 μM (IC50)

5-HT2C Receptor:1.8 μM (Ki)

References

[1]. Chagraoui A, et al. Agomelatine(S 20098) antagonizes the penile erections induced by the stimulation of 5-HT2C receptors in Wistar rats. Psychopharmacology (Berl). 2003 Oct;170(1):17-22.

 Chemical & Physical Properties

Molecular Formula C15H14D3NO3
Molecular Weight 262.32