N-Demethyl Mifepristone
Modify Date: 2024-01-11 17:38:11
N-Demethyl Mifepristone structure
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Common Name | N-Demethyl Mifepristone | ||
|---|---|---|---|---|
| CAS Number | 104004-96-8 | Molecular Weight | 415.56700 | |
| Density | 1.19g/cm3 | Boiling Point | 628.9ºC at 760mmHg | |
| Molecular Formula | C28H33NO2 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 334.1ºC | |
Use of N-Demethyl MifepristoneN-Demethyl Mifepristone (RU 42633) is an active metabolite of Mifepristone (HY-13683). The affinities of N-Demethyl Mifepristone to the glucocorticoid receptor is 61% compared with 100% for Mifepristone[1]. |
| Name | N-Demethyl Mifepristone |
|---|---|
| Synonym | More Synonyms |
| Description | N-Demethyl Mifepristone (RU 42633) is an active metabolite of Mifepristone (HY-13683). The affinities of N-Demethyl Mifepristone to the glucocorticoid receptor is 61% compared with 100% for Mifepristone[1]. |
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| Related Catalog | |
| References |
| Density | 1.19g/cm3 |
|---|---|
| Boiling Point | 628.9ºC at 760mmHg |
| Molecular Formula | C28H33NO2 |
| Molecular Weight | 415.56700 |
| Flash Point | 334.1ºC |
| Exact Mass | 415.25100 |
| PSA | 49.33000 |
| LogP | 5.45520 |
| Vapour Pressure | 1.11E-16mmHg at 25°C |
| Index of Refraction | 1.625 |
|
~88%
N-Demethyl Mife... CAS#:104004-96-8 |
| Literature: Von Geldern, Thomas W.; Tu, Noah; Kym, Philip R.; Link, James T.; Jae, Hwan-Soo; Lai, Chunqiu; Apelqvist, Theresa; Rhonnstad, Patrik; Hagberg, Lars; Koehler, Konrad; Grynfarb, Marlena; Goos-Nilsson, Annika; Sandberg, Johnny; Osterlund, Marie; Barkhem, Tomas; Hoeglund, Marie; Wang, Jiahong; Fung, Steven; Wilcox, Denise; Nguyen, Phong; Jakob, Clarissa; Hutchins, Charles; Faernegfardh, Mathias; Kauppi, Bjoern; Oehman, Lars; Jacobson, Peer B. Journal of Medicinal Chemistry, 2004 , vol. 47, # 17 p. 4213 - 4230 |
|
~76%
N-Demethyl Mife... CAS#:104004-96-8 |
| Literature: ABBOTT LABORATORIES Patent: WO2004/869 A1, 2003 ; Location in patent: Page 24; 27 ; WO 2004/000869 A1 |
|
~80%
N-Demethyl Mife... CAS#:104004-96-8 |
| Literature: Rao, Pemmaraju N.; Acosta, C. Kirk; Cessac, James W.; Bahr, Martin L.; Kim, Hyun K. Steroids, 1999 , vol. 64, # 3 p. 205 - 212 |
|
~61%
N-Demethyl Mife... CAS#:104004-96-8 |
| Literature: Mais; Chen; Wagoner; Scott Hayes; Wang Journal of Labelled Compounds and Radiopharmaceuticals, 1995 , vol. 36, # 12 p. 1199 - 1203 |
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