2687273-52-3
2687273-52-3 structure
- Name: PARP/EZH2-IN-1
- Chemical Name: PARP/EZH2-IN-1
- CAS Number: 2687273-52-3
- Molecular Formula: C43H41FN8O5
- Molecular Weight: 768.83
- Catalog: Signaling Pathways Cell Cycle/DNA Damage PARP
- Create Date: 2021-12-19 11:33:30
- Modify Date: 2025-09-15 19:22:06
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PARP/EZH2-IN-1 is a first-in-class dual PARP (IC50 6.87 nM) and EZH2 (IC50 36.51 nM) inhibitor for triple-negative breast cancer with wild-type BRCA.
| Name | PARP/EZH2-IN-1 |
|---|
| Description | PARP/EZH2-IN-1 is a first-in-class dual PARP (IC50 6.87 nM) and EZH2 (IC50 36.51 nM) inhibitor for triple-negative breast cancer with wild-type BRCA. |
|---|---|
| Related Catalog | |
| Target |
PARP-1:6.87 nM (IC50) EZH2:36.51 nM (IC50) |
| References |
| Molecular Formula | C43H41FN8O5 |
|---|---|
| Molecular Weight | 768.83 |