Name | LSN 3213128 |
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Description | LSN 3213128 is a selective, nonclassical, orally bioavailable antifolate with potent and specific inhibitory activity for aminoimidazole-4-carboxamide ribonucleotide formyltransferase (AICARFT), with IC50 of 16 nM for AICARFT enzyme inhibiton and 19 nM in cells. Anti-tumor activity[1]. |
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Related Catalog | |
Target |
IC50: 16 nM (AICARFT), 19 nM (AICARFT in cells)[1] |
References |
Molecular Formula | C17H16FN3O4S2 |
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Molecular Weight | 409.46 |