PAC1R antagonist 1
Names
[ CAS No. ]:
2305204-24-2
[ Name ]:
PAC1R antagonist 1
Biological Activity
[Description]:
PAC1R antagonist 1 (compound 3d) is a potent and orally active antagonist of PAC1 receptor. PAC1R antagonist 1 can inhibit pituitary adenylate cyclase-activating polypeptide (PACAP)- and nerve injury-induced allodynia[1].
[Related Catalog]:
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C17H17ClN6O2
[ Molecular Weight ]:
372.81