mGAT3/4-IN-2

Names

[ CAS No. ]:
2556833-68-0

[ Name ]:
mGAT3/4-IN-2

[Description]:

mGAT3/4-IN-2 (compound 27b) is a potent mGAT3/mGAT4 inhibitor, with pIC50 values of 5.44 and 5.25, respectively[1].

[Related Catalog]:

Signaling Pathways >> Membrane Transporter/Ion Channel >> GABA Receptor

Research Areas >> Metabolic Disease

Research Areas >> Neurological Disease

Signaling Pathways >> Neuronal Signaling >> GABA Receptor

[Target]

pIC50: 5.12 ± 0.08 (mGAT1), 5.14 ± 0.07 (mGAT2), 5.44 ± 0.08 (mGAT3), 5.25 ± 0.04 (mGAT4)[1]

[References]

[ Molecular Formula ]:
C₂₆H₃₂ClN₃OS₂

[ Molecular Weight ]:
502.13