TIPP

Names

[ Name ]:
TIPP

[Synonym ]:
Tyr-tic-phe-phe-OH
H-Tyr-Tic-Phe-Phe-OH
L-Phenylalanine,L-tyrosyl-L-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-L-phenylalanyl
TIPP

Biological Activity

[Description]:

TIPP is a potent and selective δ-opioid antagonist with a Ki value of 1.22 nM[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Opioid Receptor

Signaling Pathways >> Neuronal Signaling >> Opioid Receptor

Research Areas >> Neurological Disease

[References]

[1]. Schiller PW, et al. The TIPP opioid peptide family: development of delta antagonists, delta agonists, and mixed mu agonist/delta antagonists. Biopolymers. 1999;51(6):411-25.

Chemical & Physical Properties

[ Molecular Formula ]:
C₃₇H₃₈N₄O₆

[ Molecular Weight ]:
634.72

[ Exact Mass ]:
634.27900

[ PSA ]:
162.06000

[ LogP ]:
4.17510

Related Compounds

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