GLUT1-IN-2

• 常用名: GLUT1-IN-2
• 英文名: GLUT1-IN-2
• CAS号: 305357-89-5
• 分子量: 327.38
• 密度: N/A
• 沸点: N/A
• 分子式: C₂₁H₁₇N₃O
• 熔点: N/A
• 闪点: N/A

GLUT1-IN-2用途

GLUT1-IN-2(化合物17)是一种GLUT1抑制剂,IC50值为12μM。GLUT1-IN-2对恶性疟原虫己糖转运蛋白PfHT具有抑制作用,IC50值为13μM。GLUT1-IN-2可用于感染的研究[1]。

GLUT1-IN-2名称

• 英文名: Benzamide, N-[3-(1H-benzimidazol-2-yl)phenyl]-3-methyl

GLUT1-IN-2生物活性

• 描述: GLUT1-IN-2(化合物17)是一种GLUT1抑制剂,IC50值为12μM。GLUT1-IN-2对恶性疟原虫己糖转运蛋白PfHT具有抑制作用,IC50值为13μM。GLUT1-IN-2可用于感染的研究[1]。
• 相关类别:
  研究领域 >> 感染
• 靶点实验:

  IC50: 12 μM (GLUT1), 13 μM (PfHT)[1]

• 体外研究: GLUT1-IN-2(0-100μM)抑制GLUT1和PfHT的活性,IC50值分别为12和13μM[1]。

GLUT1-IN-2物理化学性质

• 分子式: C₂₁H₁₇N₃O
• 分子量: 327.38
• InChIKey: BFAZKDZNMRHORZ-UHFFFAOYSA-N
• SMILES: Cc1cccc(C(=O)Nc2cccc(-c3nc4ccccc4[nH]3)c2)c1

GLUT1-IN-2靶点实验

查看更多实验

实验名称：Antileishmanial activity against axenic amastigote Leishmania donovani MHOM/SD/1962/1... 来源：ChEMBL 靶标：Leishmania donovani External Id：CHEMBL3406137

实验名称：Antileishmanial activity against axenic amastigote Leishmania donovani MHOM/SD/1962/1... 来源：ChEMBL 靶标：Leishmania donovani External Id：CHEMBL3406135

实验名称：Antibacterial activity against Chlamydia pneumoniae CWL029 infected in human HL cells... 来源：ChEMBL 靶标：Chlamydia pneumoniae External Id：CHEMBL1286501

实验名称：Antileishmanial activity against axenic amastigote Leishmania donovani MHOM/SD/1962/1... 来源：ChEMBL 靶标：Leishmania donovani External Id：CHEMBL3406136

实验名称：Cytotoxicity against human HL cells assessed as cell viability at 10 uM after 72 hrs ... 来源：ChEMBL 靶标：HL External Id：CHEMBL1286502

实验名称：Antibacterial activity against Chlamydia pneumoniae CWL029 infected in human HL cells... 来源：ChEMBL 靶标：Chlamydia pneumoniae External Id：CHEMBL1286504

实验名称：Cytotoxicity against human HL cells at 2.5 uM after 72 hrs by celltiter-glo analysis 来源：ChEMBL 靶标：HL External Id：CHEMBL1286507

实验名称：Antibacterial activity against Staphylococcus aureus ATCC 25923 assessed as inhibitio... 来源：ChEMBL 靶标：Staphylococcus aureus External Id：CHEMBL1286508

实验名称：Antibacterial activity against Escherichia coli ATCC 25922 assessed as inhibition of ... 来源：ChEMBL 靶标：Escherichia coli External Id：CHEMBL1286509

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