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305357-89-5 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Leishmania donovani
External ID: CHEMBL3406137
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2015
Volume: 25
Issue: 9
First Page: 1933
Last Page: 1937
DOI: 10.1016/j.bmcl.2015.03.027

Target ChEMBL ID: CHEMBL367
ChEMBL Target Name: Leishmania donovani
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
Inhibition=17%
Inhibition=17%
Inhibition=22%
Inhibition=36%
InhibitionNot Determined
Inhibition=20%
Inhibition=26%
Inhibition=19%
Inhibition=26%
Inhibition=35%
Inhibition=32%
Inhibition=27%
Inhibition=32%
Inhibition=28%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Leishmania donovani
External ID: CHEMBL3406135
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2015
Volume: 25
Issue: 9
First Page: 1933
Last Page: 1937
DOI: 10.1016/j.bmcl.2015.03.027

Target ChEMBL ID: CHEMBL367
ChEMBL Target Name: Leishmania donovani
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=56%
Inhibition=83%
Inhibition=55%
Inhibition=77%
Inhibition=22%
Inhibition=56%
Inhibition=59%
Inhibition=57%
Inhibition=51%
Inhibition=64%
Inhibition=69%
Inhibition=63%
Inhibition=83%
Inhibition=97%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Chlamydia pneumoniae
External ID: CHEMBL1286501
Protocol: N/A
Comment: Journal: J Med Chem
Year: 2010
Volume: 53
Issue: 21
First Page: 7664
Last Page: 7674
DOI: 10.1021/jm1008083

Target ChEMBL ID: CHEMBL612694
ChEMBL Target Name: Chlamydia pneumoniae
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=99%
Inhibition=99%
Inhibition=99%
Inhibition=99%
Inhibition=0%
Inhibition=0%
Inhibition=98%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Leishmania donovani
External ID: CHEMBL3406136
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2015
Volume: 25
Issue: 9
First Page: 1933
Last Page: 1937
DOI: 10.1016/j.bmcl.2015.03.027

Target ChEMBL ID: CHEMBL367
ChEMBL Target Name: Leishmania donovani
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
Inhibition=43%
Inhibition=68%
Inhibition=47%
Inhibition=50%
InhibitionNot Determined
Inhibition=21%
Inhibition=52%
Inhibition=35%
Inhibition=26%
Inhibition=52%
Inhibition=50%
Inhibition=41%
Inhibition=58%
Inhibition=44%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:HL
External ID: CHEMBL1286502
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 2010
Volume: 53
Issue: 21
First Page: 7664
Last Page: 7674
DOI: 10.1021/jm1008083

Target ChEMBL ID: CHEMBL612594
ChEMBL Target Name: HL
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
Activity=98%
Activity=69%
Activity=90%
Activity=95%
Activity=96%
Activity=100%
Activity=99%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Chlamydia pneumoniae
External ID: CHEMBL1286504
Protocol: N/A
Comment: Journal: J Med Chem
Year: 2010
Volume: 53
Issue: 21
First Page: 7664
Last Page: 7674
DOI: 10.1021/jm1008083

Target ChEMBL ID: CHEMBL612694
ChEMBL Target Name: Chlamydia pneumoniae
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
GI=80%
GI=80%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:HL
External ID: CHEMBL1286507
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 2010
Volume: 53
Issue: 21
First Page: 7664
Last Page: 7674
DOI: 10.1021/jm1008083

Target ChEMBL ID: CHEMBL612594
ChEMBL Target Name: HL
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeActivity Comment
ActivityNon-toxic
ActivityNon-toxic
ActivityNon-toxic
ActivityNon-toxic
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Staphylococcus aureus
External ID: CHEMBL1286508
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 2010
Volume: 53
Issue: 21
First Page: 7664
Last Page: 7674
DOI: 10.1021/jm1008083

Target ChEMBL ID: CHEMBL352
ChEMBL Target Name: Staphylococcus aureus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
GINot Active
GI=85%
GINot Active
GINot Active
GINot Active
GINot Active
GINot Active
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL1286509
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 2010
Volume: 53
Issue: 21
First Page: 7664
Last Page: 7674
DOI: 10.1021/jm1008083

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeActivity Comment
GINot Active
GINot Active
GINot Active
GINot Active
GINot Active
GINot Active
GINot Active