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Ribociclib D6

更新时间:2024-01-12 19:11:46

Ribociclib D6结构式
Ribociclib D6结构式
品牌特惠专场
常用名 Ribociclib D6 英文名 LEE011-D6
CAS号 1328934-40-2 分子量 440.57
密度 N/A 沸点 N/A
分子式 C23H24D6N8O 熔点 N/A
MSDS N/A 闪点 N/A

 Ribociclib D6用途


Ribociclib D6 (LEE011 D6) 是 Ribociclib 的一种氘代化合物。Ribociclib 是一种高度特异性的 CDK4/6 抑制剂,IC50 值分别为 10 nM 和 39 nM,对 cyclin B/CDK1 复合体的活性低于其 1000 倍。

 Ribociclib D6名称

英文名 Ribociclib D6

 Ribociclib D6生物活性

描述 Ribociclib D6 (LEE011 D6) 是 Ribociclib 的一种氘代化合物。Ribociclib 是一种高度特异性的 CDK4/6 抑制剂,IC50 值分别为 10 nM 和 39 nM,对 cyclin B/CDK1 复合体的活性低于其 1000 倍。
相关类别
参考文献

[1]. VanArsdale T, et al. Molecular Pathways: Targeting the Cyclin D-CDK4/6 Axis for Cancer Treatment. Clin Cancer Res. 2015 Jul 1;21(13):2905-10.

 Ribociclib D6物理化学性质

分子式 C23H24D6N8O
分子量 440.57
品牌现货直购
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Ribociclib D6价格

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