常用名 | PF-05198007 | CAS号 | 1235406-19-5 |
---|---|---|---|
价格 | 纯度 | 99.0% | |
备货期 | 10天 | 库存 | 现货 |
产品详情(用途,包装等)
用途: PF-05198007 is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 9 nM, no significant activity against Nav1.5 (IC50>10 uM); increases action potential rheobase in small diameter mDRG neurons, demonstrates in vivo efficacy in a mouse capsaicin-induced neurogenic flare model. 物理化学性质: CAS号:1235406-19-5 常用中文名:PF-05198007 常用英文名:PF-05198007 分子式:C19H12ClF4N5O3S2 分子量:533.901 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |