1-Aminomethylbenzocycloalkanes: Conformationally Restricted Hallucinogenic Phenethylamine Analogues as Functionally Selective 5-HT2A Receptor Agonists 1

TH McLean, JC Parrish, MR Braden…

文献索引：Togo, Hideo; Kikuchi, Osamu Heterocycles, 1989 , vol. 28, # 1 p. 373 - 381

被引用次数: 59

摘要

... Volume: Page: Digital Object Identifier (DOI). ... (S)-2, 460 ± 53, 89 ± 1.3, >10000, >10000. 1 (“2C-B”), 27 ± 3.1, 82 ± 1.2, nd c, nd c. a IA = intrinsic activity, the percent maximal stimulation relative to 10 μM 5-HT. b Parrish et al. ...

~17%

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~17%

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~15%

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