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mAChR-IN-1

Names

[ CAS No. ]:
119391-56-9

[ Name ]:
mAChR-IN-1

[Synonym ]:
1'-(4-iodobenzyl)-3-phenyl-[3,4'-bipiperidine]-2,6-dione
mAChR-IN-1

Biological Activity

[Description]:

mAChR-IN-1 is a potent muscarinic cholinergic receptor(mAChR) antagonist with IC50 of 17 nM.

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> mAChR
Signaling Pathways >> Neuronal Signaling >> mAChR
Research Areas >> Neurological Disease

[References]

[1]. Wilson AA, et al. Synthesis and biological evaluation of [125I]- and [123I]-4-iododexetimide, a potent muscarinic cholinergic receptor antagonist. J Med Chem. 1989 May;32(5):1057-62.


[Related Small Molecules]

Carbachol | Darifenacin HBr | Arecoline hydrobromide | Pirenzepine, Dihydrochloride | Glycopyrrolate | Imidafenacin | Benztropine Mesylate | Xanomeline oxalate | Batefenterol | Bethanechol chloride | Cevimeline hydrochloride hemihydrate | Otilonium Bromide | solifenacin | VU0467154 | Anisodamine

Chemical & Physical Properties

[ Molecular Formula ]:
C23H25IN2O2

[ Molecular Weight ]:
488.36100

[ Exact Mass ]:
488.09600

[ PSA ]:
49.41000

[ LogP ]:
4.14450

[ Storage condition ]:
2-8℃

Related Compounds