Clocinnamox mesylate

Modify Date: 2024-01-11 17:21:14

Clocinnamox mesylate structure	Common Name	Clocinnamox mesylate
	CAS Number	117332-69-1	Molecular Weight	601.11
	Density	N/A	Boiling Point	753.4ºC at 760mmHg
	Molecular Formula	C₃₀H₃₃ClN₂O₇S	Melting Point	N/A
	MSDS	N/A	Flash Point	409.4ºC

Use of Clocinnamox mesylate

Clocinnamox (mesylate) is a potent opioid antagonist acting at mu, kappa and delta-receptors. Clocinnamox is a selective mu-receptor antagonist than kappa and delta-receptors[1].

Name	14b-(p-chlorocinnamoylamino)-7,8-dihydro-n-cyclopropylmethylmorphinone mesylate
Synonym	More Synonyms

Description	Clocinnamox (mesylate) is a potent opioid antagonist acting at mu, kappa and delta-receptors. Clocinnamox is a selective mu-receptor antagonist than kappa and delta-receptors[1].
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Opioid Receptor Signaling Pathways >> Neuronal Signaling >> Opioid Receptor Research Areas >> Neurological Disease
References	[1]. S D Comer, et, al. Clocinnamox: a novel, systemically-active, irreversible opioid antagonist. J Pharmacol Exp Ther. 1992, 262, 3. [2]. E R Butelman, et, al. Clocinnamox antagonism of opioid suppression of schedule-controlled responding in rhesus monkeys. Psychopharmacology (Berl). 1996, 123, 4.

Description

Clocinnamox (mesylate) is a potent opioid antagonist acting at mu, kappa and delta-receptors. Clocinnamox is a selective mu-receptor antagonist than kappa and delta-receptors[1].

Related Catalog

Signaling Pathways >> GPCR/G Protein >> Opioid Receptor

Signaling Pathways >> Neuronal Signaling >> Opioid Receptor

Research Areas >> Neurological Disease

References

[1]. S D Comer, et, al. Clocinnamox: a novel, systemically-active, irreversible opioid antagonist. J Pharmacol Exp Ther. 1992, 262, 3.

[2]. E R Butelman, et, al. Clocinnamox antagonism of opioid suppression of schedule-controlled responding in rhesus monkeys. Psychopharmacology (Berl). 1996, 123, 4.

Boiling Point	753.4ºC at 760mmHg
Molecular Formula	C₃₀H₃₃ClN₂O₇S
Molecular Weight	601.11
Flash Point	409.4ºC
Exact Mass	600.17000
PSA	141.62000
LogP	4.92970
Vapour Pressure	1.74E-23mmHg at 25°C

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Clocinnamox mesylate

Use of Clocinnamox mesylate

Names

Clocinnamox mesylate Biological Activity

Chemical & Physical Properties

Synonyms