HA-100
Modify Date: 2025-08-29 18:05:50
HA-100 structure
|
Common Name | HA-100 | ||
|---|---|---|---|---|
| CAS Number | 84468-24-6 | Molecular Weight | 277.34200 | |
| Density | 1.332g/cm3 | Boiling Point | 497.4ºC at 760 mmHg | |
| Molecular Formula | C13H15N3O2S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 254.6ºC | |
Use of HA-100HA-100 is an inhibitor of cGMP-dependent protein kinase (PKG), cAMP-dependent protein kinase (PKA), Protein kinase C (PKC) and MLC-kinase with IC50s of 4, 8, 12 and 240 μM, respectively. |
| Name | 5-piperazin-1-ylsulfonylisoquinoline |
|---|---|
| Synonym | More Synonyms |
| Description | HA-100 is an inhibitor of cGMP-dependent protein kinase (PKG), cAMP-dependent protein kinase (PKA), Protein kinase C (PKC) and MLC-kinase with IC50s of 4, 8, 12 and 240 μM, respectively. |
|---|---|
| Related Catalog | |
| Target |
PKC:12 μM (IC50) PKG:4 μM (IC50) PKA:8 μM (IC50) MLCK:240 μM (IC50) |
| References |
| Density | 1.332g/cm3 |
|---|---|
| Boiling Point | 497.4ºC at 760 mmHg |
| Molecular Formula | C13H15N3O2S |
| Molecular Weight | 277.34200 |
| Flash Point | 254.6ºC |
| Exact Mass | 277.08800 |
| PSA | 70.68000 |
| LogP | 2.17620 |
| Index of Refraction | 1.639 |
| InChIKey | UPTYCYWTFGTCCG-UHFFFAOYSA-N |
| SMILES | O=S(=O)(c1cccc2cnccc12)N1CCNCC1 |
| Storage condition | −20°C |
| HS Code | 2935009090 |
|---|---|
| Summary | 2935009090 other sulphonamides VAT:17.0% Tax rebate rate:9.0% Supervision conditions:none MFN tariff:6.5% General tariff:35.0% |
| Tocris-0543 |
| ha-100 |
| MFCD01310980 |