ARC 239 dihydrochloride

Modify Date: 2025-08-27 02:32:31

ARC 239 dihydrochloride Structure
ARC 239 dihydrochloride structure
 Common Name ARC 239 dihydrochloride
CAS Number 55974-42-0 Molecular Weight 480.42700
Density N/A Boiling Point N/A
Molecular Formula C24H31Cl2N3O3 Melting Point N/A
MSDS Chinese Flash Point N/A

 Use of ARC 239 dihydrochloride


ARC 239 dihydrochloride is a selective α2B/2C adrenoceptor antagonist (pKd values are 5.95, 7.41 and 7.56 at α2A, α2B, and α2C receptors respectively). ARC 239 dihydrochloride binds to CHO cell membranes expressing human recombinant a2A-, a2B- or a2C-adrenoceptor subtypes with pKis of 5.6, 8.4, and 7.08, respectively[1].

 Names

Name 2-{2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl}-4,4-dimethyl-1,3(2 H,4H)-isoquinolinedione dihydrochloride
Synonym More Synonyms

 ARC 239 dihydrochloride Biological Activity

Description ARC 239 dihydrochloride is a selective α2B/2C adrenoceptor antagonist (pKd values are 5.95, 7.41 and 7.56 at α2A, α2B, and α2C receptors respectively). ARC 239 dihydrochloride binds to CHO cell membranes expressing human recombinant a2A-, a2B- or a2C-adrenoceptor subtypes with pKis of 5.6, 8.4, and 7.08, respectively[1].
Related Catalog
Target

Alpha-2B adrenergic receptor

5-HT1A Receptor

References

[1]. M R Corboz, et al. Pharmacological characterization of alpha 2-adrenoceptor-mediated responses in pig nasal mucosa. Auton Autacoid Pharmacol. 2003 Aug;23(4):208-19.

 Chemical & Physical Properties

Molecular Formula C24H31Cl2N3O3
Molecular Weight 480.42700
Exact Mass 479.17400
PSA 53.09000
LogP 4.32220

 Synonyms

Pertussis Toxin
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