SIS3
Modify Date: 2024-01-02 09:33:22
SIS3 structure
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Common Name | SIS3 | ||
|---|---|---|---|---|
| CAS Number | 521984-48-5 | Molecular Weight | 489.993 | |
| Density | N/A | Boiling Point | 737.2ºC at 760 mmHg | |
| Molecular Formula | C28H28ClN3O3 | Melting Point | N/A | |
| MSDS | Chinese USA | Flash Point | 399.7ºC | |
Use of SIS3SIS3 is a cell-permeable and selective inhibitor of Smad3. It inhibits Smad3 phosphorylation with an IC50 of 3 µM. |
| Name | sis3 |
|---|---|
| Synonym | More Synonyms |
| Description | SIS3 is a cell-permeable and selective inhibitor of Smad3. It inhibits Smad3 phosphorylation with an IC50 of 3 µM. |
|---|---|
| Related Catalog | |
| References |
| Boiling Point | 737.2ºC at 760 mmHg |
|---|---|
| Molecular Formula | C28H28ClN3O3 |
| Molecular Weight | 489.993 |
| Flash Point | 399.7ºC |
| Exact Mass | 489.181915 |
| PSA | 56.59000 |
| LogP | 5.59550 |
| Storage condition | -20℃ |
| Personal Protective Equipment | Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter |
|---|---|
| RIDADR | NONH for all modes of transport |
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| (2E)-1-(6,7-Dimethoxy-3,4-dihydro-2(1H)-isoquinolinyl)-3-(1-methyl-2-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)-2-propen-1-one hydrochloride (1:1) |
| 2-Propen-1-one, 1-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-3-(1-methyl-2-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)-, (2E)-, hydrochloride (1:1) |