BMS-684
Modify Date: 2024-03-07 22:56:57
BMS-684 structure
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Common Name | BMS-684 | ||
|---|---|---|---|---|
| CAS Number | 313552-29-3 | Molecular Weight | 454.52 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C27H26N4O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of BMS-684BMS-684 is a selective DGKα inhibitor with an IC50 of 15 nM. BMS-684 inhibits DGKα kinase activity with >100-fold selectivity over the related DGK type I family members DGKβ and DGKγ. BMS-684 does not inhibit any of the other seven DGK isozymes[1]. |
| Name | BMS-684 |
|---|
| Description | BMS-684 is a selective DGKα inhibitor with an IC50 of 15 nM. BMS-684 inhibits DGKα kinase activity with >100-fold selectivity over the related DGK type I family members DGKβ and DGKγ. BMS-684 does not inhibit any of the other seven DGK isozymes[1]. |
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| Related Catalog | |
| Target |
IC50: 15 nM (DGKα)[1] |
| References |
| Molecular Formula | C27H26N4O3 |
|---|---|
| Molecular Weight | 454.52 |
| InChIKey | XIVOLEKHEMYRBO-UHFFFAOYSA-N |
| SMILES | Cn1c(=O)c([N+](=O)[O-])c(N2CCN(C(c3ccccc3)c3ccccc3)CC2)c2ccccc21 |