SJ1461
Modify Date: 2024-01-02 19:44:30
SJ1461 structure
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Common Name | SJ1461 | ||
|---|---|---|---|---|
| CAS Number | 2924546-70-1 | Molecular Weight | 484.00 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C21H18ClN7OS2 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of SJ1461SJ1461 is a potent and orally active BET inhibitor. SJ1461 inhibits BRD2 (BD1), and BRD2 (BD2), BRD4 (BD1), and BRD4 (BD2) with IC50 values of 1.6 nM, 0.1 nM, 6.5 nM, and 0.2 nM, respectively[1]. |
| Name | SJ1461 |
|---|
| Description | SJ1461 is a potent and orally active BET inhibitor. SJ1461 inhibits BRD2 (BD1), and BRD2 (BD2), BRD4 (BD1), and BRD4 (BD2) with IC50 values of 1.6 nM, 0.1 nM, 6.5 nM, and 0.2 nM, respectively[1]. |
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| Related Catalog | |
| Target |
BRD2 (BD1):1.6 nM (IC50) BRD2 (BD2):0.1 nM (IC50) BRD4 (BD1):6.5 nM (IC50) BRD4 (BD2):0.2 nM (IC50) |
| References |
| Molecular Formula | C21H18ClN7OS2 |
|---|---|
| Molecular Weight | 484.00 |